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- Mossine, Andrew
V.; Brooks, Allen F.; Makaravage, Katarina J.; Miller, Jason M.; Ichiishi, Naoko; Sanford, Melanie S.; Scott, Peter J. H.
- Organic letters 2015 v.17 no.23 pp. 5780-5783
- acids; boronic acids; chemical reactions; moieties; organic compounds
- ... A copper-mediated radiofluorination of aryl- and vinylboronic acids with K¹⁸F is described. This method exhibits high functional group tolerance and is effective for the radiofluorination of a range of electron-deficient, -neutral, and -rich aryl-, heteroaryl-, and vinylboronic acids. This method has been applied to the synthesis of [¹⁸F]FPEB, a PET radiotracer for quantifying metabotropic glutama ...
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